Preserved supervised synthesis

Retatrutide synthesis · version 2

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Supervised synthesis

What do selected human studies report about Retatrutide?

Manually reviewed September 15, 2026 · version 2

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Three selected reports cover early retatrutide studies and the later TRANSCEND-T2D-1 phase 3 diabetes trial. Populations, comparators and primary endpoints differ across the studies.123

Bottom line from this bounded source set

Selected trials reported weight reduction and improved glycated hemoglobin. The newer phase 3 diabetes study supports a glycemic effect in its studied population, but these reports do not establish prevention of long-term complications; gastrointestinal adverse events and discontinuations matter.123

Reviewed study record

Phase 2 obesity trial

Design

A double-blind, randomized, placebo-controlled Phase 2 trial followed participants for 48 weeks and assessed body-weight change and safety.1

Population

The trial enrolled 338 adults with obesity, or overweight plus at least one weight-related condition.1

Outcomes reported

At 48 weeks, reported mean body-weight change ranged from -8.7% to -24.2% across retatrutide groups, compared with -2.1% for placebo. Gastrointestinal events were the most common adverse events, and heart-rate increases peaked at 24 weeks before declining.1

Limitations

This was a sponsor-funded Phase 2 trial with 48-week follow-up; it was not a long-term cardiovascular-outcomes or rare-harms study.1

Reviewed study record

Phase 2 type 2 diabetes trial

Design

A randomized, double-blind, placebo- and active-comparator-controlled Phase 2 trial evaluated glycated hemoglobin at 24 weeks and body weight at 36 weeks.2

Population

The trial randomized 281 adults with type 2 diabetes and elevated body-mass index at 42 U.S. centers; 275 were included in efficacy analyses.2

Outcomes reported

At 24 weeks, reported glycated-hemoglobin changes ranged from -0.43 to -2.02 percentage points across retatrutide groups, compared with -0.01 for placebo and -1.41 for the active comparator. Reported body-weight change at 36 weeks ranged from -3.19% to -16.94% across retatrutide groups.2

Limitations

The sponsor-funded trial had 36-week follow-up, 79% completed treatment, and 84% of participants were White; those features limit conclusions about durability and generalizability.2

Reviewed study record

TRANSCEND-T2D-1: phase 3 diabetes study

Design

A blinded randomized placebo-controlled trial assessed 40-week glycated hemoglobin change under NCT06354660.3

Population

The trial randomized 537 adults with type 2 diabetes inadequately controlled with diet and exercise alone.3

Outcomes reported

Under the treatment-regimen analysis, HbA1c decreased by 1.69–1.94 percentage points across active groups versus 0.81 with placebo. Gastrointestinal events were common; adverse-event discontinuations occurred in 2–5% of active groups and none of the placebo group.3

Limitations

HbA1c and weight changes do not establish prevention of long-term complications. The report recorded two deaths in one active group, which the authors considered unrelated to study treatment; it reported no severe hypoglycemia.3

Reviewed source set

  1. PubMed · 37366315Triple-Hormone-Receptor Agonist Retatrutide for Obesity - A Phase 2 Trial ↗PubMed PMID 37366315 · EFetch XML reviewed 2026-08-18 · payload SHA-256 167232d6f5d1818faabbc3d98c283b2ffad85563d5e10720f8e23347bba1ad1b
    No registered Crossref update in the reviewed snapshotChecked August 19, 2026 for DOI 10.1056/nejmoa2301972. This bounded result is not proof that the publication has never been corrected or retracted. Open the pinned Crossref work endpoint ↗
  2. PubMed · 37385280Retatrutide, a GIP, GLP-1 and glucagon receptor agonist, for people with type 2 diabetes: a randomised, double-blind, placebo and active-controlled, parallel-group, phase 2 trial conducted in the USA ↗PubMed PMID 37385280 · EFetch XML reviewed 2026-08-18 · payload SHA-256 766a11f2d979da96a8a2b79353159b0e0472215d1e391b8f8f5d09a142c5fdcd
    No registered Crossref update in the reviewed snapshotChecked August 19, 2026 for DOI 10.1016/s0140-6736(23)01053-x. This bounded result is not proof that the publication has never been corrected or retracted. Open the pinned Crossref work endpoint ↗
  3. PubMed · 42250575Efficacy and safety of retatrutide, a GIP, GLP-1, and glucagon receptor agonist, in people with type 2 diabetes and inadequate glycaemic control with diet and exercise (TRANSCEND-T2D-1): a double-blind, randomised, phase 3 trial. ↗PubMed PMID 42250575 · EFetch XML reviewed 2026-09-15 · payload SHA-256 c7b0d7e8d9f2053a0083809311fa312b449f6271b7cde41ea747e8bdf0a318c4
    No registered Crossref update in the reviewed snapshotChecked September 15, 2026 for DOI 10.1016/s0140-6736(26)00967-0. This bounded result is not proof that the publication has never been corrected or retracted. Open the pinned Crossref work endpoint ↗